2-Methoxyestrone
Cat. No.：YN370689
| 产品名称: | 2-Methoxyestrone |
| CAS No.: | 362-08-3 |
| Chemical Name: | 3-hydroxy-2-methoxy-estra-1,3,5(10)-trien-17-one |
| Synonyms: | |
| 分子量: | 300.39 |
| 分子式: | C₁₉H₂₄O₃ |
| SMILES: | C[C@]1([C@](CC2)([H])[C@]3([H])CCC4=C(C=C(OC)C(O)=C4)[C@@]3([H])CC1)C2=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | 2-Methoxyestrone 是一种甲氧基苯二酚雌激素，也是雌酮的代谢物，其 pKa 值为 10.81。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
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Fotsis, T., Zhang, Y., Pepper, M.S., et al.The endogenous oestrogen metabolite 2-methoxyoestradiol inhibits angiogenesis and suppresses tumour growthNature368(6468),237-239(1994)
Seeger, H., Mueck, A.O., and Lippert, T.H.Effect of estradiol metabolites on prostacyclin synthesis in human endothelial cell culturesLife Sci.65(13),PL167-PL170(1999)
Liu, D., and Bachmann, K.A.An investigation of the relationship between estrogen, estrogen metabolites and blood cholesterol levels in ovariectomized ratsJ. Pharmacol. Exp. Ther.286(1),561-568(1998)
