IRL 2500
Cat. No.:YN320263
CAS No. :169545-27-1
产品名称: | IRL 2500 |
CAS No.: | 169545-27-1 |
Chemical Name: | |
Synonyms: | |
分子量: | 573.68 |
分子式: | C₃₆H₃₅N₃O₄ |
SMILES: | O=C(O)[C@H](CC1=CNC2=CC=CC=C12)NC([C@@H](CC3=CC=C(C4=CC=CC=C4)C=C3)N(C(C5=CC(C)=CC(C)=C5)=O)C)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | IRL 2500 是一种有效的内皮素受体 (Endothelin receptor) 拮抗剂,其 ETB和 ETA受体的IC50值分别为 1.3 和 94 nM。 IRL 2500 在体内抑制 ETB 受体介导的血压升高和肾血管阻力。 |
IC50和靶点: | [{name:"ETB:1.3 nM (IC50)"},{name: "ETA:94 nM (IC50)"}] |
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Clinical Trial: | |
Solvent & Solubility: |