Y06137
Cat. No.:YN310115
CAS No. :2226534-49-0
产品名称: | Y06137 |
CAS No.: | 2226534-49-0 |
Chemical Name: | |
Synonyms: | |
分子量: | 444.57 |
分子式: | C₂₇H₃₂N₄O₂ |
SMILES: | CC1=NOC(C1=C2)=CC=C2C3=NC(C=C4)=C(N3CC5CCCCC5)C=C4N6CCOC[C@@H]6C |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Y06137 是一种有效的选择性BET抑制剂,与BRD4(1)溴结构域结合,Kd值为 81 nM。Y06137 用于研究去势抵抗性前列腺癌 (CRPC)。 |
IC50和靶点: | [{name:"BRD4(1):81 nM (Kd)"}] |
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Clinical Trial: | |
Solvent & Solubility: |