BAY1238097
Cat. No.:YN310123
CAS No. :1564268-08-1
产品名称: | BAY1238097 |
CAS No.: | 1564268-08-1 |
Chemical Name: | |
Synonyms: | BAY1238097 |
分子量: | 451.56 |
分子式: | C₂₅H₃₃N₅O₃ |
SMILES: | O=C(N1N=C(C2=CC=C(N3CCN(C)CC3)C=C2)C4=CC(OC)=C(OC)C=C4C[C@@H]1C)NC |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | BAY1238097 是一种有效的、BET 与组蛋白结合的选择性抑制剂,通过下调c-Myc水平及下游转录组,在AML (急性髓性白血病) 和MM (多发性骨髓瘤) 模型中表现出较强的抗增殖活性 (IC50值 <100 nM)。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |