TP-238
Cat. No.：YN310138
| 产品名称: | TP-238 |
| CAS No.: | 2415263-04-4 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 458.58 |
| 分子式: | C₂₂H₃₀N₆O₃S |
| SMILES: | CN(C)CCCOC1=CC=C(C=C1)C2=CC(NCCCN3N=CC=C3)=NC(S(=O)(C)=O)=N2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | TP-238 是一种有效的选择性的CECR2/BPTF双探针，pIC50值分别为 7.5 和 6.5。TP-238 还抑制 BRD9，pIC50为 5.9，对其他 338 种激酶的活性较低。 |
| IC50和靶点: | [{name:"CECR2:7.5 (pIC50)"},{name: "BRD9:5.9 (pIC50)"},{name: "CECR2:30 nM (IC50)"},{name: "CECR2:10 nM (Kd)"},{name: "BPTF:6.5 (pIC50)"},{name: "BPTF:350 nM (IC50)"},{name: "BPTF:120 nM (Kd)"}] |
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| Solvent & Solubility: |
