Molibresib
Cat. No.:YN310207
CAS No. :1260907-17-2
产品名称: | Molibresib |
CAS No.: | 1260907-17-2 |
Chemical Name: | (S)-2-(6-(4-chlorophenyl)-8-methoxy-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)-N-ethylacetamide |
Synonyms: | I-BET762; GSK525762; GSK525762A |
分子量: | 423.90 |
分子式: | C₂₂H₂₂ClN₅O₂ |
SMILES: | ClC1=CC=C(C2=N[C@@H](CC(NCC)=O)C3=NN=C(C)N3C4=CC=C(OC)C=C24)C=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Molibresib (I-BET762; GSK525762) 是BET 溴结构域抑制剂,IC50为32.5-42.5 nM。 |
IC50和靶点: | |
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