Bromosporine
Cat. No.:YN310282
CAS No. :1619994-69-2
产品名称: | Bromosporine |
CAS No.: | 1619994-69-2 |
Chemical Name: | ethyl (3-methyl-6-(4-methyl-3-(methylsulfonamido)phenyl)-[1,2,4]triazolo[4,3-b]pyridazin-8-yl)carbamate |
Synonyms: | Bromosporine;Carbamic acid, N-[3-methyl-6-[4-methyl-3-[(methylsulfonyl)amino]phenyl]-1,2,4-triazolo[4,3-b]pyridazin-8-yl]-, ethyl ester;Bromorsporine;Bioomosporine;GTPL8234;C17H20N6O4S;Bromosporine, >=98% (HPLC);AOB6807;HMS3653C21;2286AH;s7233;AK175193;A4 |
分子量: | 404.44 |
分子式: | C₁₇H₂₀N₆O₄S |
SMILES: | O=C(OCC)NC1=CC(C2=CC=C(C)C(NS(=O)(C)=O)=C2)=NN3C1=NN=C3C |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Bromosporine对于BRD2,BRD4,BRD9和CECR2的IC50分别为410nM、290nM、122nM和17nM。 |
IC50和靶点: | |
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Clinical Trial: | |
Solvent & Solubility: |
Gallenkamp, D., Gelato, K.A., Haendler, B., et al.Bromodomains and their pharmacological inhibitorsChem. Med. Chem.9(3),438-464(2014)