Velusetrag hydrochloride
Cat. No.:YN380449
| 产品名称: | Velusetrag hydrochloride |
| CAS No.: | 866933-51-9 |
| Chemical Name: | |
| Synonyms: | TD-5108 hydrochloride |
| 分子量: | 541.104 |
| 分子式: | C25H37ClN4O5S |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Velusetrag (TD-5108) hydrochloride 是一种具有口服活性,有效和选择性的血清素5-HT4受体 (5-HT4R) 激动剂,pKi为 7.7。Velusetrag hydrochloride 对 5-HT2A和 5-HT2B受体没有亲和力 (Ki>10 μM)。Velusetrag hydrochloride 可用于胃肠道疾病和帕金森病的研究。 |
| IC50和靶点: | [{name:"5-HT4 Receptor:7.7 (pKi)"}] |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |