PD173074
Cat. No.：YN440076
CAS No. ：219580-11-7
规格
价格(RMB)
库存
| 产品名称: | PD173074 |
| CAS No.: | 219580-11-7 |
| Chemical Name: | N-[2-[[4-(diethylamino)butyl]amino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-N'-(1,1-dimethylethyl)-urea |
| Synonyms: | PD173074, PD 173074 |
| 分子量: | 523.67 |
| 分子式: | C₂₈H₄₁N₇O₃ |
| SMILES: | O=C(NC1=NC2=NC(NCCCCN(CC)CC)=NC=C2C=C1C3=CC(OC)=CC(OC)=C3)NC(C)(C)C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PD173074 是有效的FGFR1抑制剂，IC50为 25 nM；也可抑制VEGFR2的活性，IC50值为 100-200 nM，对 FGFR1 的活性是 PDGFR 和 c-Src 的1000多倍。 |
| IC50和靶点: | [{name:"FGFR1:25 nM (IC50)"},{name: "VEGFR2:100 nM (IC50)"}] |
| In Vitro: | |
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| Clinical Trial: | |
| Solvent & Solubility: |
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