HTH-01-091
Cat. No.:YN270691
产品名称: | HTH-01-091 |
CAS No.: | 2000209-42-5 |
Chemical Name: | |
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分子量: | 499.43 |
分子式: | C26H28Cl2N4O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | HTH-01-091 是一种强效且选择性的maternal embryonic leucine zipper kinase (MELK)抑制剂,其IC50为 10.5 nM。HTH-01-091 还能抑制PIM1/2/3、RIPK2、DYRK3、smMLCK和CLK2。HTH-01-091 可用于乳腺癌研究。 |
IC50和靶点: | [{name:"DYRK4:41.8 nM (IC50)"},{name: "PIM1:60.6 nM (IC50)"},{name: "mTOR:632 nM (IC50)"},{name: "CDK7:1230 nM (IC50)'}, 'PIM2', 'PIM3'] |
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