MX1013
Cat. No.:YN270766
CAS No. :582316-00-5
产品名称: | MX1013 |
CAS No.: | 582316-00-5 |
Chemical Name: | 5-fluoro-3-[[(2S)-3-methyl-1-oxo-2-[[(phenylmethoxy)carbonyl]amino]butyl]amino]-4-oxo-pentanoic acid |
Synonyms: | CV1013; Z-VD-FMK |
分子量: | 382.3835032 |
分子式: | C18H23FN2O6 |
SMILES: | O=C(O)CC(NC([C@@H](NC(OCC1=CC=CC=C1)=O)C(C)C)=O)C(CF)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MX1013 是一种有效的、不可逆的二肽caspase抑制剂,具有抗细胞凋亡活性。MX1013 抑制重组人caspase 3,IC50为 30 nM。 |
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Yang, W., Guastella, J., Huang, J.-C., et al.MX1013, a dipeptide caspase inhibitor with potent in vivo antiapoptotic activityBr. J. Pharmacol.140(2),402-412(2003)