SKF89976A hydrochloride
Cat. No.:YN360014
产品名称: | SKF89976A hydrochloride |
CAS No.: | 85375-15-1 |
Chemical Name: | 1-(4,4-Diphenyl-3-butenyl)-3-piperidinecarboxylic Acid Hydrochloride; |
Synonyms: | d,l |
分子量: | 371.90 |
分子式: | C₂₂H₂₆ClNO₂ |
SMILES: | O=C(C1CN(CC/C=C(C2=CC=CC=C2)/C3=CC=CC=C3)CCC1)O.[H]Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | SKF89976A hydrochloride 是一种选择性GABA转运蛋白GAT-1抑制剂,作用于 CHO 细胞中的 GAT-1,GAT-2 和 GAT-3,IC50分别为 0.28 μM,137.34 μM 和 202.8 μM。 |
IC50和靶点: | |
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Jinzenji, A., et al.: J. Pharmacol. Sci., 125, 217-226 (2014)
Sunol, C., et al.: Neurochem. Res., 35, 1384-1390 (2010)