Tracazolate hydrochloride
Cat. No.：YN360888
CAS No. ：1135210-68-2
| 产品名称: | Tracazolate hydrochloride |
| CAS No.: | 1135210-68-2 |
| Chemical Name: | |
| Synonyms: | ICI 136753 hydrochloride |
| 分子量: | 340.85 |
| 分子式: | C₁₆H₂₅ClN₄O₂ |
| SMILES: | O=C(C1=C(C)N=C(N(CC)N=C2)C2=C1NCCCC)OCC.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Tracazolate (ICI 136753) hydrochloride 是一种有效的GABAA受体调节剂。Tracazolate hydrochloride 对 β3 具有选择性，同时增强 α1β1γ2s (EC50=13.2μM) 和 α1β3γ2 (EC50=1.5 μM)。Tracazolate hydrochloride 的效力 (EC50) 是由受体复合物中的第三亚基 (γ1-3, δ, ε) 的性质决定。Tracazolate hydrochloride 具有抗焦虑和抗惊厥活性。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
