Ibutamoren Mesylate
Cat. No.:YN321286
CAS No. :159752-10-0
产品名称: | Ibutamoren Mesylate |
CAS No.: | 159752-10-0 |
Chemical Name: | 2-amino-N-[(1R)-2-[1,2-dihydro-1-(methylsulfonyl)spiro[3H-indole-3,4'-piperidin]-1'-yl]-2-oxo-1-[(phenylmethoxy)methyl]ethyl]-2-methyl-propanamide, methanesulfonate |
Synonyms: | 伊布莫仑甲磺酸盐; MK-677; MK-0677 |
分子量: | 624.77 |
分子式: | C₂₈H₄₀N₄O₈S₂ |
SMILES: | CC(N)(C(N[C@@H](C(N1CCC2(CN(C3=C2C=CC=C3)S(=O)(C)=O)CC1)=O)COCC4=CC=CC=C4)=O)C.CS(=O)(O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Ibutamoren Mesylate (MK-677) 是一种有效的,非肽段类生长激素促分泌素受体 (GHSR) 激动剂。Ibutamoren Mesylate 是一种有效的,具有口服活性的生长激素 (GH) 促分泌素。 |
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Kojima, M., Hosoda, H., Date, Y., et al.Ghrelin is a growth-hormone-releasing acylated peptide from stomachNature402(6762),656-660(1999)
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Smith, R.G., Pong, S.S., Hickey, G., et al.Modulation of pulsatile GH release through a novel receptor in hypothalamus and pituitary glandRecent Prog. Horm. Res.51,261-286(1996)
Patchett, A.A., Nargund, R.P., Tata, J.R., et al.Design and biological activities of L-163,191 (MK-0677): A potent, orally active growth hormone secretagogueProc. Natl. Acad. Sci. USA92(15),7001-7005(1995)