Leuprolide Acetate
Cat. No.：YN320783
CAS No. ：74381-53-6
| 产品名称: | Leuprolide Acetate |
| CAS No.: | 74381-53-6 |
| Chemical Name: | 6-D-leucine-9-(N-ethyl-L-prolinamide)-1-9-luteinizing hormone-releasing factor (swine), monoacetate |
| Synonyms: | Leuprorelin acetate |
| 分子量: | 1269.45 |
| 分子式: | C₆₁H₈₈N₁₆O₁₄ |
| SMILES: | CC(O)=O.O=C(N[C@@H](CO)C(N[C@H](C(N[C@H](CC(C)C)C(N[C@@H](CC(C)C)C(N[C@@H](CCCNC(N)=N)C(N(CCC1)[C@@H]1C(NCC)=O)=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)[C@@H](NC([C@@H](NC([C@@H](N3)CCC3=O)=O)CC4=CN=CN4)=O)CC5=CNC6=C5C=CC=C6 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Leuprolide Acetate (Leuprorelin acetate) 是一种促性腺激素释放激素 (GnRH) 类似物，能作为 GnRH 受体 (GnRH receptor) 激动剂。Leuprolide Acetate 可用于前列腺癌、子宫内膜异位症、子宫肌瘤、中枢性早熟、多发性硬化症的研究。Leuprolide Acetate 能改善大鼠模型中的实验性自身免疫性脑脊髓炎 (EAE)。 |
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Plosker, G.L., and Brogden, R.N.Leuprorelin. A review of its pharmacology and therapeutic use in prostatic cancer, endometriosis and other sex hormone-related disordersDrugs.48(6),930-967(1994)
Gravel, P., Samland, D., Löffler, M., et al.Two innovative pharmaceutical forms of leuprorelin: results from 818 patients with advanced prostate cancerAdv. Ther.30(3),271-285(2013)
