Alarelin Acetate
Cat. No.:YN321130
CAS No. :79561-22-1
产品名称: | Alarelin Acetate |
CAS No.: | 79561-22-1 |
Chemical Name: | 6-D-alanine-9-(N-ethyl-L-prolinamide)-1-9-luteinizing hormone-releasing factor (swine), diacetate |
Synonyms: | Alarelin |
分子量: | 1287.42 |
分子式: | C₆₀H₈₆N₁₆O₁₆ |
SMILES: | O=C(N[C@@H](CO)C(N[C@@H](CC1=CC=C(O)C=C1)C(N[C@H](C)C(N[C@@H](CC(C)C)C(N[C@@H](CCCNC(N)=N)C(N2CCC[C@H]2C(NCC)=O)=O)=O)=O)=O)=O)[C@@H](NC([C@@H](NC([C@@H](N3)CCC3=O)=O)CC4=CN=CN4)=O)CC5=CNC6=CC=CC=C65.CC(O)=O.CC(O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Alarelin acetate是合成的GnRH激动剂。 |
IC50和靶点: | |
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Han, Y.-G., Kang, S.S., Seong, J.Y., et al.Negative regulation of gonadotropin-releasing hormone and gonadotropin-releasing hormone receptor gene expression by a gonadotrophin-releasing hormone agonist in the rat hypothalamusJ. Neuroendocrinol.11(3),195-201(1999)
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Xiaoying, X., and Sanyuan, Z.Effect of alarelin acetate on human endometrial carcinoma in nude mice transplantation tumor and expression of POT1Zhonghua Linchuang Yishi Zazhi9(7),63-66(2015)