Iperoxo
Cat. No.：YN322428
CAS No. ：247079-84-1
| 产品名称: | Iperoxo |
| CAS No.: | 247079-84-1 |
| Chemical Name: | 4-[(4,5-dihydro-3-isoxazolyl)oxy]-N,N,N-trimethyl-2-butyn-1-aminium, monoiodide |
| Synonyms: | |
| 分子量: | 324.15873 |
| 分子式: | C10H17N2O2 • I |
| SMILES: | C[N+](C)(C)CC#CCOC1=NOCC1.[I-] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Iperoxo 是一种有效的毒蕈碱乙酰胆碱受体 (mAChR) 的超级激动剂。[3H]Iperoxo 可用于直接探测毒蕈碱受体的激活相关构象转变。 |
| IC50和靶点: | |
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Croy, C.H., Schober, D.A., Xiao, H., et al.Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M2 and M4 receptorsMol. Pharmacol.86(1),106-115(2014)
Dallanoce, C., Conti, P., De Amici, M., et al.Synthesis and functional characterization of novel derivatives related to oxotremorine and oxotremorine-MBioorg. Med. Chem.7(8),1539-1547(1999)
Barocelli, E., Ballabeni, V., Bertoni, S., et al.Evidence for specific analgesic activity of a muscarinic agonist selected among a new series of acetylenic derivativesLife Sci.68(15),1775-1785(2001)
