CDK12-IN-E9
Cat. No.:YN290154
| 产品名称: | CDK12-IN-E9 |
| CAS No.: | 2020052-55-3 |
| Chemical Name: | |
| Synonyms: | E9;CDK12-IN-E9 |
| 分子量: | 434.53 |
| 分子式: | C₂₄H₃₀N₆O₂ |
| SMILES: | C=CC(NC1=CC=CC(NC2=CC(N3[C@H](CCO)CCCC3)=NC4=C(CC)C=NN24)=C1)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CDK12-IN-E9 是一种有效的选择性共价CDK12抑制剂和非共价CDK9抑制剂,同时避免了 ABC 转运蛋白介导的外排。CDK12-IN-E9 对 CDK7/CyclinH 复合物的结合能力较弱,IC50> 1 μM。 |
| IC50和靶点: | |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |