Pergolide mesylate
Cat. No.：YN1730060
CAS No. ：66104-23-2
| 产品名称: | Pergolide mesylate |
| CAS No.: | 66104-23-2 |
| Chemical Name: | 8β-[(methylthio)methyl]-6-propyl-ergoline, monomethanesulfonate |
| Synonyms: | 甲磺酸培高利特; Pergolide methanesulfonate; LY127809 |
| 分子量: | 410.59 |
| 分子式: | C₂₀H₃₀N₂O₃S₂ |
| SMILES: | [H][C@@]1(N(CCC)C[C@H](CSC)C[C@@]12[H])CC3=CNC4=CC=CC2=C43.CS(=O)(O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Pergolide mesylate 是有抗帕金森病特性的多巴胺受体激动剂。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
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Zhang, X.X., Jin, G.Z., and Wei, Y.F.Agonistic actions of pergolide on firing activity of dopamine neurons in substantia nigra compacta areaZhongguo Yao Li Xue Bao.16(5),423-427(1995)
Yoshimura, N., Mizuta, E., Yoshida, O., et al.Therapeutic effects of dopamine D1/D2 receptor agonists on detrusor hyperreflexia in 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine-lesioned parkinsonian cynomolgus monkeysJ. Pharmacol. Exp. Ther.286(1),228-233(1998)
Bendele, A.M., Spaethe, S.M., Benslay, D.N., et al.Anti-inflammatory activity of pergolide, a dopamine receptor agonistJ. Pharmacol. Exp. Ther.259(1),169-175(1991)
