GLP-26
Cat. No.:YN250348
CAS No. :2133017-36-2
产品名称: | GLP-26 |
CAS No.: | 2133017-36-2 |
Chemical Name: | |
Synonyms: | GLP-26,GLP 26,GLP26 |
分子量: | 373.35 |
分子式: | C₁₉H₁₇F₂N₃O₃ |
SMILES: | O=C(C1=C(C)C(C(C(NCC#C)=O)=O)=C(C)N1C)NC2=CC=C(F)C(F)=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GLP-26 是一种HBV衣壳组装调节剂 (CAM),抑制 Hep AD38 系统中的 HBV DNA 复制 (IC50=3 nM), 并在 1 μM 时使 cccDNA 降低> 90%。GLP-26 破坏前基因组 RNA 的衣壳化,导致核衣壳解体,并减少 cccDNA 库。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |