Cilobradine hydrochloride
Cat. No.:YN360663
产品名称: | Cilobradine hydrochloride |
CAS No.: | 186097-54-1 |
Chemical Name: | 3-[[(3S)-1-[2-(3,4-dimethoxyphenyl)ethyl]-3-piperidinyl]methyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one, monohydrochloride |
Synonyms: | DK-AH 269 |
分子量: | 519.07 |
分子式: | C₂₈H₃₉ClN₂O₅ |
SMILES: | O=C1N(C[C@@H]2CN(CCC3=CC=C(OC)C(OC)=C3)CCC2)CCC4=CC(OC)=C(OC)C=C4C1.[H]Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Cilobradine是一种HCN通道阻断剂。 |
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Stieber, J., Wieland, K., Stöckl, G., et al.Bradycardic and proarrhythmic properties of sinus node inhibitorsMol. Pharmacol.69(4),1328-1337(2006)
Bois, P., Chatelier, A., Bescond, J., et al.Pharmacology of hyperpolarization-activated cyclic nucleotide-gated (HCN) channelsIon channels and their inhibitors,33-51(2011)