MS417
Cat. No.：YN250189
CAS No. ：916489-36-6
| 产品名称: | MS417 |
| CAS No.: | 916489-36-6 |
| Chemical Name: | |
| Synonyms: | GTPL7512 |
| 分子量: | 414.91 |
| 分子式: | C₂₀H₁₉ClN₄O₂S |
| SMILES: | O=C(OC)C[C@H]1C2=NN=C(C)N2C3=C(C(C)=C(C)S3)C(C4=CC=C(Cl)C=C4)=N1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | MS417 是一种选择性的 BET 特异性蛋白BRD4的抑制剂，能够与 BRD4-BD1 和 BRD4-BD2 结合，IC50值分别为 30，46 nM，Kd值分别为 36.1，25.4 nM; MS417 对 CBP BRD 的选择性较低，IC50值为 32.7 μM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
