ESI-08
Cat. No.:YN322825
CAS No. :301177-43-5
产品名称: | ESI-08 |
CAS No.: | 301177-43-5 |
Chemical Name: | |
Synonyms: | |
分子量: | 353.48 |
分子式: | C20H23N3OS |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ESI-08 是一种有效的选择性EPAC拮抗剂,可以完全抑制EPAC1和EPAC2(IC50为 8.4 μM) 的活性。ESI-08 选择性阻断 cAMP 诱导的EPAC激活,但不抑制 cAMP 介导的PKA激活。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |