Imetit dihydrobromide
Cat. No.：YN320103
| 产品名称: | Imetit dihydrobromide |
| CAS No.: | 32385-58-3 |
| Chemical Name: | carbamimidothioic acid, 2-(1H-imidazol-5-yl)ethyl ester, dihydrobromide |
| Synonyms: | VUF 8325 dihydrobromide; SKF 91105 dihydrobromide |
| 分子量: | 332.06 |
| 分子式: | C₆H₁₂Br₂N₄S |
| SMILES: | NC(SCCC1=CN=CN1)=N.Br.Br |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Imetit dihydrobromide (VUF 8325 dihydrobromide) 是组胺H3和H4受体的高亲和力的强激动剂，Ki值分别为 0.3 和 2.7 nM。Imetit dihydrobromide 模拟组胺对嗜酸性粒细胞形状改变的作用 (EC50=25 nM)。 |
| IC50和靶点: | [{name:"H3 Receptor:0.3 nM (Ki)"},{name: "H4 receptor:2.7 nM (Ki)"}] |
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