Pitolisant
Cat. No.:YN320560
CAS No. :362665-56-3
产品名称: | Pitolisant |
CAS No.: | 362665-56-3 |
Chemical Name: | 1-[3-[3-(4-Chlorophenyl)propoxy]propyl]piperidine; 3-(4-Chlorophenyl)propyl 3-piperidinopropyl Ether; Wakix; |
Synonyms: | Tiprolisant |
分子量: | 295.85 |
分子式: | C₁₇H₂₆ClNO |
SMILES: | ClC1=CC=C(CCCOCCCN2CCCCC2)C=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Pitolisant 是一种有效的选择性的非咪唑类重组人组胺H3受体反相激动剂,Ki为 0.16 nM。 |
IC50和靶点: | |
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Harwell, V., et al.: Medicines, 7, 55 (2020)
Imeri, F., et al.: Neuropharmacology, 186, 108464 (2021)
Li, S., et al.: Expert Rev. Clin. Pharmacol., 13, 79 (2020)