Rupatadine D4 fumarate
Cat. No.：YN320746
| 产品名称: | Rupatadine D4 fumarate |
| CAS No.: | 1795153-63-7 |
| Chemical Name: | 8-Chloro-6,11-dihydro-11-[1-[(5-methyl-3-pyridinyl)methyl]-4-piperidinylidene-d4]- 5H-benzo[5,6]cyclohepta[1,2-b]pyridine (2E)-2-Butenedioate; Rupafin-d4 Fumarate; |
| Synonyms: | UR-12592 D4 fumarate |
| 分子量: | 536.05 |
| 分子式: | C₃₀H₂₆D₄ClN₃O₄ |
| SMILES: | CC1=CN=CC(CN2C([2H])([2H])C/C(CC2([2H])[2H])=C3C4=CC=C(Cl)C=C4CCC5=CC=CN=C5\3)=C1.OC(/C=C/C(O)=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Rupatadine D4 fumarate (UR-12592 D4 fumarate) 是Rupatadine fumarate 的氘代标记物。Rupatadine Fumarate (UR-12592 Fumarate) 富马酸盐是PAF/H1受体双抑制剂，Ki值分别为0.55 μM 和 0.1 μM。 |
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| Solvent & Solubility: |
Merlos, M., et al.: J. Pharmacol. Exp. Ther., 280, 114 (1997), Guadano, E.M., et al.: Allergy, 59, 766 (2004),
