Oxomemazine
Cat. No.：YN320780
| 产品名称: | Oxomemazine |
| CAS No.: | 3689-50-7 |
| Chemical Name: | 10-[3-(Dimethylamino)-2-methylpropyl]phenothiazine 5,5-Dioxide; 6487 RP; 6847 RP; Doxergan |
| Synonyms: | |
| 分子量: | 330.44 |
| 分子式: | C₁₈H₂₂N₂O₂S |
| SMILES: | CC(CN1C2=C(C=CC=C2)S(C3=CC=CC=C13)(=O)=O)CN(C)C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体 (histamine H1-receptor) 阻滞剂，具有明显的抗毒蕈碱活性。Oxomemazine 是毒菌碱 M1 受体的选择性拮抗剂，在高 (histamine H1-receptor=84 nM, M1受体) 和低 (histamine H1-receptor=1.65 μM, M2受体) 亲和力位点上显示了 20 倍的差异。Oxomemazine 是一种用于咳嗽研究相关研究的一种抗组胺和抗胆碱能试剂。 |
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Meindl, W. et al.: Archiv der Pharmazie , Vol.322, P: 133-6 (1989)
