Chlorprothixene hydrochloride
Cat. No.：YN321441
CAS No. ：6469-93-8
| 产品名称: | Chlorprothixene hydrochloride |
| CAS No.: | 6469-93-8 |
| Chemical Name: | (3Z)-3-(2-chloro-9H-thioxanthen-9-ylidene)-N,N-dimethyl-1-propanamine, monohydrochloride |
| Synonyms: | chlorprothixene HCI |
| 分子量: | 352.32 |
| 分子式: | C₁₈H₁₉Cl₂NS |
| SMILES: | CN(C)CC/C=C1C2=C(SC3=C\1C=CC=C3)C=CC(Cl)=C2.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Chlorprothixene hydrochloride 是一种多巴胺 (dopamine) 和组胺 (histamine) 受体拮抗剂，高亲和力地结合人 D1，D2，D3，D5，H1 受体，Ki分别为 18 nM，2.96 nM，4.56 nM，9 nM 和 3.75 nM。具有抗精神病作用。 |
| IC50和靶点: | [{name:"Human D1 Receptor:18 nM (Ki)"},{name: "Human D2 Receptor:2.96 nM (Ki)"},{name: "Human D3 Receptor:4.56 nM (Ki)"},{name: "Human D5 Receptor:9 nM (Ki)"},{name: "Human H1 Receptor:3.75 nM (Ki)"}] |
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