Betahistine dihydrochloride
Cat. No.：YN321523
| 产品名称: | Betahistine dihydrochloride |
| CAS No.: | 5579-84-0 |
| Chemical Name: | N-methyl-2-pyridineethanamine, dihydrochloride |
| Synonyms: | 盐酸倍他司汀 |
| 分子量: | 209.12 |
| 分子式: | C₈H₁₄Cl₂N₂ |
| SMILES: | CNCCC1=CC=CC=N1.Cl.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Betahistine dihydrochloride 是一种口服有效的组胺 H1 受体 (histamine H1 receptor) 激动剂和 H3 受体 (H1 receptor) 的拮抗剂。Betahistine dihydrochloride 用于类风湿性关节炎 (RA) 的研究。 |
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Timmerman, H.Histamine agonists and antagonistsActa Otolaryngol. Suppl.479,5-11(1991)
Bertlich, M., Ihler, F., Sharaf, K., et al.Betahistine metabolites, aminoethylpyridine, and hydroxyethylpyridine increase cochlear blood flow in guinea pigs in vivoInt. J. Audiol.53(10),753-759(2014)
Bertlich, M., Ihler, F., Weiss, B.G., et al.Role of capillary pericytes and precapillary arterioles in the vascular mechanism of betahistine in a guinea pig inner ear modelLife Sci.187,17-21(2017)
Lian, J., Huang, X.-F., Pai, N., et al.Ameliorating antipsychotic-induced weight gain by betahistine: Mechanisms and clinical implicationsPharmacol. Res.106,51-63(2016)
