Promethazine hydrochloride
Cat. No.:YN321578
产品名称: | Promethazine hydrochloride |
CAS No.: | 58-33-3 |
Chemical Name: | N,N,α-trimethyl-10H-phenothiazine-10-ethanamine, monohydrochloride |
Synonyms: | 盐酸异丙嗪 |
分子量: | 320.88 |
分子式: | C₁₇H₂₁ClN₂S |
SMILES: | CC(N(C)C)CN1C(C=CC=C2)=C2SC3=CC=CC=C13.[H]Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Promethazine hydrochloride 是一代抗组胺药物,H1 受体强效拮抗剂和 mAChR 拮抗剂,对 5-HT2A、5-HT2C、D2和_alpha_1-adrenergic受体也有一定的亲和性。 |
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Tsay, M.E., Procopio, G., Anderson, B.D., et al.Abuse and intentional misuse of promethazine reported to US Poison Centers: 2002 to 2012J. Addict. Med.9(3),233-237(2015)
Lynch, K.L., Shapiro, B.J., Coffa, D., et al.Promethazine use among chronic pain patientsDrug Alcohol Depend.,92-97(2015)