MK-0249
Cat. No.:YN322020
产品名称: | MK-0249 |
CAS No.: | 862309-06-6 |
Chemical Name: | |
Synonyms: | |
分子量: | 431.45 |
分子式: | C₂₃H₂₄F₃N₃O₂ |
SMILES: | O=C1N(C2=CC=C(OCCCN3CCCC3)C=C2)C(C)=NC4=C1C(C(F)(F)F)=CC=C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MK-0249 是一种有效的histamine H3 受体拮抗剂,对人体 H3 受体的Ki值为 1.7 nM。 |
IC50和靶点: | [{name:"human H3 receptor:1.7 nM (IC50)"},{name: "rhesus H3 receptor:4.3 nM (Ki)"},{name: "human H3 receptor:6.8 nM (Ki)"},{name: "rat H3 receptor:33 nM (Ki)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |