CPI-169
Cat. No.:YN310288
CAS No. :1802175-07-0
产品名称: | CPI-169 |
CAS No.: | 1802175-07-0 |
Chemical Name: | |
Synonyms: | CPI 169 R-enantiomer |
分子量: | 528.66 |
分子式: | C₂₇H₃₆N₄O₅S |
SMILES: | CC(N1)=CC(OC)=C(CNC(C2=C(C)N([C@H](C)C3CCN(S(=O)(CC)=O)CC3)C4=CC=CC=C24)=O)C1=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CPI-169 (CPI 169 R-enantiomer) 是一种新颖的,有效的EZH2抑制剂,能够抑制 EZH2 WT,EZH2 Y641N 和 EZH1 的活性,IC50值分别为 0.24 nM,0.51 nM 和 6.1 nM。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |