KDM5A-IN-1
Cat. No.：YN310001
CAS No. ：1905481-36-8
| 产品名称: | KDM5A-IN-1 |
| CAS No.: | 1905481-36-8 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 290.36 |
| 分子式: | C₁₅H₂₂N₄O₂ |
| SMILES: | O=C(C1CC1)N[C@@H]2CCN(C(C3=CC(C(C)C)=NN3)=O)C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | KDM5A-IN-1 是一种有效的，口服可生物利用的泛组氨酸赖氨酸脱甲基酶 5KDM5抑制剂，对KDM5A，KDM5B和KDM5C的IC50值分别为 45 nM，56 nM 和 55 nM，对 PC9 H3K4Me3 的EC50值为 960 nM。KDM5A-IN-1 对其他KDM酶 (1A，2B，3B，4C，6A，7B) 的效力明显较低。 |
| IC50和靶点: | |
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