LPA2 antagonist 1
Cat. No.:YN321173
CAS No. :1017606-66-4
产品名称: | LPA2 antagonist 1 |
CAS No.: | 1017606-66-4 |
Chemical Name: | N-[(1S)-2-[4-[(3,4-dichlorophenyl)sulfonyl]-1-piperazinyl]-1-methylethyl]-7-methyl-thieno[3,2-d]pyrimidin-4-amine |
Synonyms: | |
分子量: | 500.46 |
分子式: | C₂₀H₂₃Cl₂N₅O₂S₂ |
SMILES: | ClC1=C(Cl)C=C(S(=O)(N2CCN(C[C@@H](NC3=NC=NC4=C3SC=C4C)C)CC2)=O)C=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | LPA2 antagonist 1是LPA2的拮抗剂,IC50值为17 nM。 |
IC50和靶点: | |
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Clinical Trial: | |
Solvent & Solubility: |
Beck, H.P., Kohn, T., Rubenstein, S., et al.Discovery of potent LPA2 (EDG4) antagonists as potential anticancer agentsBioorg. Med. Chem. Lett.18(3),1037-1041(2008)