Tipelukast
Cat. No.:YN320934
产品名称: | Tipelukast |
CAS No.: | 125961-82-2 |
Chemical Name: | 4-[6-acetyl-3-[3-[(4-acetyl-3-hydroxy-2-propylphenyl)thio]propoxy]-2-propylphenoxy]-butanoic acid |
Synonyms: | KCA 757; MN 001 |
分子量: | 530.67 |
分子式: | C₂₉H₃₈O₇S |
SMILES: | CC(C1=C(O)C(CCC)=C(SCCCOC2=C(CCC)C(OCCCC(O)=O)=C(C(C)=O)C=C2)C=C1)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Tipelukast (KCA 757) 是一种白三烯受体 (leukotriene receptor) 拮抗剂,是一种可口服的抗炎剂,同时可用于哮喘的研究。 |
IC50和靶点: | [{name:"LTD4:6.41 (pA2, In guinea-pigs)"},{name: "LTE4:6.45 (pA2, In guinea-pigs)"}] |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |
Rajasekaran, M., Locke, K.W., and Parsons, C.L.MN-001, a novel oral anti-inflammatory agent, suppresses bladder hyperactivity in a rat modelBJU Int.98(2),430-434(2006)