Bremelanotide Acetate
Cat. No.：YN321193
| 产品名称: | Bremelanotide Acetate |
| CAS No.: | 1607799-13-2 |
| Chemical Name: | N-acetyl-L-norleucyl-L-α-aspartyl-L-histidyl-D-phenylalanyl-L-arginyl-L-tryptophyl-L-lysine (2→7)-lactam, monoacetate |
| Synonyms: | PT-141 Acetate |
| 分子量: | 1085.22 |
| 分子式: | C₅₂H₇₂N₁₄O₁₂ |
| SMILES: | O=C(N[C@](CCCCNC(C[C@@H]1NC([C@@H](NC(C)=O)CCCC)=O)=O)([H])C(O)=O)[C@@H](NC([C@@H](NC([C@@](NC([C@@H](NC1=O)CC2=CN=CN2)=O)([H])CC3=CC=CC=C3)=O)CCCNC(N)=N)=O)CC4=CNC5=CC=CC=C45.OC(C)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Bremelanotide Acetate (PT-141 Acetate)，α-MSH 的合成肽类似物，是黑素皮质素受体 (melanocortin receptors)，包括 MC3R 和 MC4R 的激动剂，有潜力用于性功能障碍的研究。 |
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Molinoff, P.B., Shadiack, A.M., Earle, D., et al.PT-141: A melanocortin agonist for the treatment of sexual dysfunctionAnn. N. Y. Acad. Sci.994(1),96-102(2003)
Pfaus, J., Giuliano, F., and Gelez, H.Bremelanotide: An overview of preclinical CNS effects on female sexual functionJ. Sex Med.4(Suppl 4),269-279(2007)
