4-P-PDOT
Cat. No.：YN320059
CAS No. ：134865-74-0
| 产品名称: | 4-P-PDOT |
| CAS No.: | 134865-74-0 |
| Chemical Name: | N-(1,2,3,4-tetrahydro-4-phenyl-2-naphthalenyl)-propanamide |
| Synonyms: | 4-phenyl-2- propionamidotetralin |
| 分子量: | 279.38 |
| 分子式: | C₁₉H₂₁NO |
| SMILES: | CCC(NC1CC2=C(C=CC=C2)C(C3=CC=CC=C3)C1)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | 4-P-PDOT 是一种有效的，选择性的和亲和性的褪黑激素受体 (MT2) 拮抗剂。4-P-PDOT 对MT2的选择性是 MT1 的 300 倍以上。4-P-PDOT 可显着抵消褪黑激素介导的抗氧化作用 (GSH/GSSG比，ERK 磷酸化，Nrf2 核易位，Nrf2 DNA 结合活性)。 |
| IC50和靶点: | |
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