Tasimelteon
Cat. No.：YN320915
CAS No. ：609799-22-6
| 产品名称: | Tasimelteon |
| CAS No.: | 609799-22-6 |
| Chemical Name: | N-[[(1R,2R)-2-(2,3-dihydro-4-benzofuranyl)cyclopropyl]methyl]-propanamide |
| Synonyms: | 他司美琼; BMS-214778; VEC-162 |
| 分子量: | 245.32 |
| 分子式: | C₁₅H₁₉NO₂ |
| SMILES: | [H][C@]1(C2=C3C(OCC3)=CC=C2)[C@@](CNC(CC)=O)([H])C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Tasimelteon (BMS-214778) 是一种具有口服活性，选择性的双重褪黑激素受体激动剂 (DMRA)。Tasimelteon 对 MT2 受体的亲和力是 MT1 受体的 2.1-4.4 倍。Tasimelteon 是一种昼夜节律性调节剂，具有用于非 24 小时睡眠/觉醒障碍 (Non-24) 的潜力。 |
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Lavedan, C., Forsberg, M., and Gentile, A.J.Tasimelteon: A selective and unique receptor binding profileNeuropharmacology91,142-147(2015)
