7,8-Didehydrocimigenol
Cat. No.:YN470059
产品名称: | 7,8-Didehydrocimigenol |
CAS No.: | 247923-29-1 |
Chemical Name: | 2-[[4-[2-[[[(2,4-difluorophenyl)amino]carbonyl]heptylamino]ethyl]phenyl]thio]-2-methyl-propanoic acid |
Synonyms: | GW9578; GW 9578; GW-9578. |
分子量: | 492.6 |
分子式: | C26H34F2N2O3S |
SMILES: | CCCCCCCN(CCc1ccc(cc1)SC(C)(C)C(=O)O)C(=O)Nc1ccc(F)cc1F |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GW9578 是一种亚型选择性的PPARα激动剂 (对鼠和人 PPAR-α 的EC50分别为 5 和 50 nM),具有有效的降脂活性。 |
IC50和靶点: | [{name:"mouse PPARα:5 nM (EC50)"},{name: "h-PPARα:50 nM (EC50)"}] |
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