LY456236
Cat. No.:YN322477
产品名称: | LY456236 |
CAS No.: | 338736-46-2 |
Chemical Name: | 6-Methoxy-N-(4-methoxyphenyl)-4-quinazolinamine Hydrochloride; MPMQ; |
Synonyms: | LY456236 HCl; LY456236 Hydrochloride; LY456236 ; LY 456236 ; LY-456236. |
分子量: | 317.77 |
分子式: | C16H16ClN3O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | LY456236 是一种选择性、非竞争性和具有口服活性的mGlu1受体拮抗剂,可抑制磷酸肌醇水解,其IC50为 0.145 μM。LY456236 还能抑制EGFR,IC50为 0.91 μM。 |
IC50和靶点: | |
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Solvent & Solubility: |
Shannon, H. et al.: Neuropharmacol., 49, 188 (2005)
Varty, G. et al.: Psychopharmacol., 179, 207 (2005)