Atamestane
Cat. No.：YN470076
| 产品名称: | Atamestane |
| CAS No.: | 182133-25-1 |
| Chemical Name: | 2-(4-Methoxyphenyl)-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]-benzo[b]thiophene-6-ol; LY 353381 |
| Synonyms: | LY353381; SERM III |
| 分子量: | 475.60 |
| 分子式: | C28H29NO4S |
| SMILES: | OC1=CC=C(C(OC2=CC=C(OCCN3CCCCC3)C=C2)=C(C4=CC=C(OC)C=C4)S5)C5=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Arzoxifene (LY353381) 是一种具有口服活性的选择性雌激素受体调节剂，具有类似 raloxifene 的固定环结构。Arzoxifene 对乳腺癌和子宫内膜有较强的抗雌激素作用，副作用小，对骨和脂质的雌激素有同样强的有利作用。 |
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| Solvent & Solubility: |
Suh, N., et al.: Cancer Res, 61, 8412 (2001)
Morello, K., et al.: Clinical Pharmacokinetics, 42, 361 (2003)
