Elacestrant
Cat. No.：YN470079
CAS No. ：722533-56-4
| 产品名称: | Elacestrant |
| CAS No.: | 722533-56-4 |
| Chemical Name: | |
| Synonyms: | RAD1901 |
| 分子量: | 458.63 |
| 分子式: | C30H38N2O2 |
| SMILES: | O(C([H])([H])[H])C1C([H])=C([H])C(=C(C=1[H])N(C([H])([H])C([H])([H])[H])C([H])([H])C1C([H])=C([H])C(C([H])([H])C([H])([H])N([H])C([H])([H])C([H])([H])[H])=C([H])C=1[H])[C@@]1([H])C([H])([H])C2C([H])=C([H])C(=C([H])C=2C([H])([H])C1([H])[H])O[H] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Elacestrant (RAD1901) 是一种具有口服活性的选择性estrogen receptor(ER) 降解剂 (SERD)，对ERα和ERβ的IC50值分别为 48 和 870 nM。Elacestrant 还能有效抑制 ER+乳腺癌细胞系在体内外的生长。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
