BI-0115
Cat. No.:YN1720151
CAS No. :4929-23-1
产品名称: | BI-0115 |
CAS No.: | 4929-23-1 |
Chemical Name: | |
Synonyms: | |
分子量: | 287.74 |
分子式: | C15H14ClN3O |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | BI-0115 是LOX-1的选择性抑制剂(IC50=5.4 µM),阻止细胞摄取氧化低密度脂蛋白。BI-0115 结合通过形成同二聚体配体结合域的二聚体触发受体抑制。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |
Schmidt, G.: U.S. (1968), US 3406168 A