GKI-1
Cat. No.:YN480071
产品名称: | GKI-1 |
CAS No.: | 2444764-03-6 |
Chemical Name: | |
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分子量: | 269.73 |
分子式: | C₁₅H₁₂ClN₃ |
SMILES: | ClC(C=C1)=CC=C1NC2=CC(C3=CNN=C3)=CC=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GKI-1是Greatwall (GWL)激酶抑制剂,抑制hGWLFL和hGWL-KinDom的IC50分别为4.9 和 2.5 µM。GKI-1 可高效抑制ROCK1,IC50为11 µM, 仅微弱抑制 PKA。 |
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