Gefitinib impurity 2
Cat. No.：YN480080
CAS No. ：246512-44-7
规格
价格(RMB)
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| 产品名称: | Gefitinib impurity 2 |
| CAS No.: | 246512-44-7 |
| Chemical Name: | 2-Amino-4-methoxy-5-(3-morpholinopropoxy)benzamide; Gefitinib Impurity 1 |
| Synonyms: | |
| 分子量: | 309.36 |
| 分子式: | C₁₅H₂₃N₃O₄ |
| SMILES: | O=C(N)C1=CC(OCCCN2CCOCC2)=C(OC)C=C1N |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Gefitinib impurity 2 是 Gefitinib 的杂质。Gefitinib (HY-50895) 是一种有效的，具有口服活性的选择性EGFR酪氨酸激酶抑制剂，IC50为 33 nM。Gefitinib 选择性抑制 EGF 刺激的肿瘤细胞生长 (IC50为 54 nM)，并阻断 EGF 刺激的肿瘤细胞中EGFR自磷酸化。Gefitinib 还可诱导细胞自噬 (autophagy)。Gefitinib 具有抗肿瘤活性。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
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