Dilazep dihydrochloride
Cat. No.：YN480097
CAS No. ：20153-98-4
规格
价格(RMB)
库存
| 产品名称: | Dilazep dihydrochloride |
| CAS No.: | 20153-98-4 |
| Chemical Name: | 3,4,5-trimethoxy-benzoic acid, 1,1′-[(tetrahydro-1H-1,4-diazepine-1,4(5H)-diyl)di-3,1-propanediyl] ester |
| Synonyms: | |
| 分子量: | 677.61 |
| 分子式: | C₃₁H₄₆Cl₂N₂O₁₀ |
| SMILES: | O=C(C1=CC(OC)=C(OC)C(OC)=C1)OCCCN2CCN(CCCOC(C3=CC(OC)=C(OC)C(OC)=C3)=O)CCC2.Cl.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Dilazep dihydrochloride 是腺苷摄取的抑制剂。Dilazep dihydrochloride 通过增强腺苷的作用而具有脑和冠状血管舒张作用。Dilazep dihydrochloride 还可抑制缺血性损伤，血小板聚集和核苷的膜转运。 |
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Playa, H., Lewis, T.A., Ting, A., et al.Dilazep analogues for the study of equilibrative nucleoside transporters 1 and 2 (ENT1 and ENT2)Bioorg. Med. Chem. Lett.24(24),5801-5804(2014)
Tonini, M., Perucca, E., Manzo, L., et al.Dilazep: An inhibitor of adenosine uptake with intrinsic calcium antagonistic propertiesJ. Pharm. Pharmacol.35(7),434-439(1983)
Marzilli, M., Trivella, M.G., Levantesi, D., et al.Effect of dilazep on coronary and systemic circulationsPharmacology31(2),82-87(1985)
Sumiyoshi, A., and Hayashi, T.The inhibitory effect of dilazep on in vivo accumulation of platelets onto the damaged aorta in Rabbit. II. Morphological analysisComparative Study29(1),37-42(1983)
