Dabigatran etexilate mesylate
Cat. No.:YN480227
产品名称: | Dabigatran etexilate mesylate |
CAS No.: | 872728-81-9 |
Chemical Name: | N-[[2-[[[4-[[[(hexyloxy)carbonyl]amino]iminomethyl]phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-β-alanine, methanesulfonate ethyl ester |
Synonyms: | 甲磺酸达比加群酯; BIBR 1048MS; Dabigatran etexilate methanesulfonate |
分子量: | 723.84 |
分子式: | C₃₅H₄₅N₇O₈S |
SMILES: | O=C(N(C1=NC=CC=C1)CCC(OCC)=O)C2=CC=C3C(N=C(N3C)CNC4=CC=C(C(NC(OCCCCCC)=O)=N)C=C4)=C2.CS(=O)(O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Dabigatran etexilate mesylate (BIBR 1048MS) 是具有口服活性的 Dabigatran 前药。Dabigatran etexilate mesylate 具有抗凝作用,可以预防心房颤动引起的静脉血栓栓塞和中风。 |
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Yang, X.-Z., Diao, X.-J., Yang, W.-H., et al.Design, synthesis and antithrombotic evaluation of novel dabigatran prodrugs containing methyl ferulateBioorg. Med. Chem. Lett.23(7),2089-2092(2013)