KRN5
Cat. No.:YN480515
产品名称: | KRN5 |
CAS No.: | 1800465-47-7 |
Chemical Name: | |
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分子量: | 459.47 |
分子式: | C₂₇H₂₂FNO₅ |
SMILES: | COC1=C(OC)C2=C(C=C1)C(CC3=CC=CC=C3F)=C4N(C2=O)CCC(C4=C5)=CC6=C5OCO6 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | KRN5 是 KRN2 的衍生物,是具有口服活性的T 细胞激活核因子 (NFAT5)的抑制剂,IC50值为 750 nM。KRN5 有潜力用于 NFAT5-介导的慢性关节炎的研究。 |
IC50和靶点: | |
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Clinical Trial: | |
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