MID-1
Cat. No.:YN480639
产品名称: | MID-1 |
CAS No.: | 312608-54-1 |
Chemical Name: | |
Synonyms: | ChemBridge5655896;MID 1;MID1 |
分子量: | 293.30 |
分子式: | C₁₂H₁₁N₃O₄S |
SMILES: | O=C(NC1=NC=C([N+]([O-])=O)S1)C2=CC=C(OCC)C=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MID-1 是一种 MG53-IRS-1 (Mitsugumin 53-胰岛素受体底物 1) 相互作用的抑制剂。 MID-1 破坏了 MG53 与 IRS-1 的分子缔合,并消除了 MG53 诱导的 IRS-1 泛素化和骨骼肌降解,从而导致 IRS-1 表达水平升高,胰岛素信号传导和葡萄糖摄取增加。 |
IC50和靶点: | |
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Clinical Trial: | |
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