KSC-34
Cat. No.:YN480676
产品名称: | KSC-34 |
CAS No.: | 2226201-97-2 |
Chemical Name: | |
Synonyms: | PDIA1 inhibitor KSC-34 |
分子量: | 429.95 |
分子式: | C₂₁H₂₈ClN₇O |
SMILES: | O=C(NCCNC1=NC(N(C)CCCCC2=CC=CC=C2)=NC(NCC#C)=N1)CCl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | KSC-34 是PDIA1的强效位点选择性抑制剂。KSC-34 对 a 结构域的选择性比 a' 结构域高 30 倍,并且对 PDIA1 还原酶活性具有时间依赖性。KSC-34 在复杂蛋白质组中对 PDIA 表现出选择性。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |